- Okere, C.E; & Ohabughiro, N.B.
- DOI: 10.5281/zenodo.21858285
- SSR Journal of Medical Sciences (SSRJMS)
This study
investigated the phenotypic resistance patterns, molecular determinants of
extended-spectrum β-lactamase production, phytochemical composition, and
antibacterial potential of Ocimum gratissimum leaf extracts against
extended-spectrum β-lactamase producing multidrug resistance Salmonella
isolates recovered from swine. A total of 81 Salmonella isolates were recovered
from porcine samples and identified using standard microbiological techniques.
Antimicrobial susceptibility profiling was performed using the Kirby–Bauer disc
diffusion method against ten commonly prescribed antibiotics. Extended-spectrum
β-lactamase production was phenotypically confirmed using the double-disc
synergy test, while multiplex polymerase chain reaction was employed to detect
clinically relevant β-lactamase resistance genes. Crude aqueous and ethanolic
leaf extracts of Ocimum gratissimum were prepared and evaluated for
antibacterial activity against confirmed extended-spectrum β-lactamase
producing isolates using the agar well diffusion assay. Minimum inhibitory
concentrations were determined by standard broth dilution techniques, and
qualitative phytochemical analysis was conducted by gas chromatography-mass
spectrometry to identify the major bioactive constituents responsible for
antimicrobial activity. The findings revealed a high prevalence of multidrug
resistance among the Salmonella isolates, characterized by extensive resistance
to β-lactam antibiotics and molecular confirmation of extended-spectrum
β-lactamase associated resistance genes. Both aqueous and ethanolic extracts of
Ocimum gratissimum exhibited pronounced inhibitory activity against all tested
multidrug resistance extended-spectrum β-lactamase producing isolates, with an
average Minimum inhibitory concentration of 1.78 mg/mL, demonstrating
broad-spectrum antibacterial efficacy. Phytochemical analysis confirmed the
presence of biologically active secondary metabolites, including flavonoids,
alkaloids, tannins, and saponins, whose synergistic interactions are likely
responsible for the observed antimicrobial effects. The combined phenotypic,
molecular, and phytochemical evidence highlights the remarkable therapeutic
potential of Ocimum gratissimum as a natural antimicrobial agent against
drug-resistant Salmonella. This study provides compelling evidence supporting
the development of Ocimum gratissimum which has some antimicrobial potential
against multidrug resistance and extended-spectrum β-lactamase producing
Salmonella isolates. Ocimum gratissimum can to an extent serve as a
phytotherapeutic compounds for managing infections caused by multidrug
resistance and extended spectrum β-latamase producing Salmonella within
veterinary and public health settings. Further studies involving bioactive
compound isolation, toxicity assessment, pharmacokinetic evaluation, and in
vivo efficacy are recommended to facilitate its translation into clinically
relevant antimicrobial therapeutics.
Keywords: Antimicrobial
resistance, Extended-spectrum β-lactamase, Multidrug-resistant Salmonella,
Ocimum gratissimum, Phytotherapy, Swine.
