- Ose Precious Akaniyere*, Ologhaguo Macstephen Adienbo & Austin A Ajah
- DOI: 10.5281/zenodo.19983209
- SSR Journal of Medical Sciences (SSRJMS)
The increasing global burden of neurodegenerative diseases such as Alzheimer’s disease has intensified the search for effective, plant-based therapies. Annona muricata (soursop) is a tropical plant traditionally used for various ailments, yet its neurotherapeutic potential remains underexplored. This study evaluated the cognitive-enhancing and neuroprotective properties of Annona muricata leaf extracts using a combination of phytochemical analysis, molecular docking, and behavioral testing. Phytochemical screening revealed the presence of key bioactive compounds, including flavonoids, alkaloids, glycosides, and saponins, with n-hexane extracting the highest total phytochemical yield at 45.5%, compared to 31.8% each for hydromethanol and methanol. Molecular docking showed that luteolin and quercetin exhibited strong binding affinities to critical neurological targets, including acetylcholinesterase (−12.0 docking score, −66.6%), NMDA receptors (−9.1 docking score, −50.5%), muscarinic M1 receptors (−11.7 docking score, −65%), and dopamine receptors (up to −10.8 docking score, −60%), suggesting a multi-target mechanism of neuroprotection. In vivo behavioral assessment using the Barnes Maze test demonstrated that rats treated with 300 mg/kg of Annona muricata extract significantly improved spatial learning and memory, with reductions in escape latency by up to 48.2% and in some weeks exceeding control group performance. These findings suggest that Annona muricata possesses promising neurotherapeutic potential and may serve as a natural multi-target agent in the management of Alzheimer’s disease.

